SCHEMBL9701385

SCHEMBL9701385

NN1CC(CN2CCCNCC2)Oc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 3/20 0.48
ADRA2A P08913 2/20 0.48
ADRA2B P18089 2/20 0.48
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
SCN1A P35498 1/20 0.48
SCN2A Q99250 1/20 0.48
SCN3A Q9NY46 1/20 0.48
HRH3 Q9Y5N1 2/20 0.46
HTR1A P08908 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
CXCR4 P61073 5/20 0.38
MEN1 O00255 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CCR2 P41597 1/20 0.38
CXCL12 P48061 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701550 0.88 ADRA2A (0.60) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9701487 0.88 ADRA2A (0.56) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9701405 0.87 ADRA2A (0.62) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9699307 0.82 ADRA2C (0.45) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL2546786 0.81 ADRA2A (0.74) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9700324 0.80 ADRA2A (0.47) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9700145 0.79 ADRA2A (0.46) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9701310 0.79 HRH3 (0.50) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL9700525 0.76 HTR1A (0.47) ADRA2CADRA2AADRA2BADRA1DADRA1A
SCHEMBL6985659 0.74 ADRA2A (0.73) ADRA2CADRA2AADRA2BADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed