SCHEMBL9701537

SCHEMBL9701537

Cc1cc2cc(Cl)cc3c2n1C(CN1CCCC1)CO3

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
SCN1A P35498 1/20 0.34
SCN2A Q99250 1/20 0.34
SCN3A Q9NY46 1/20 0.34
CNR1 P21554 5/20 0.33
CNR2 P34972 5/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C9 P11712 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 3/20 0.32
MAPT P10636 1/20 0.32
NPC1 O15118 1/20 0.32
MTOR P42345 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699289 0.97 CNR1 (0.33) HRH3ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9701612 0.90 HRH3 (0.39) HRH3CNR1CNR2CYP3A4CYP2C9
SCHEMBL9728633 0.89 L3MBTL1 (0.36) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701569 0.81 CNR1 (0.34) HRH3ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9700209 0.80 CNR1 (0.46) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699311 0.74 ADRB1 (0.32) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9700282 0.74 HRH3 (0.41) HRH3ADRA2AADRA2BADRA2CCNR1
SCHEMBL8069945 0.72 CNR1 (0.56) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9700318 0.68 CNR1 (0.51) CNR1CNR2CYP3A4CYP2C9MEN1
SCHEMBL9701634 0.66 DRD2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed