SCHEMBL9701697

SCHEMBL9701697

COP(=O)(Cc1nc2cc(C)c(C)cc2nc1CBr)OC

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.44
NQO2 P16083 5/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 2/20 0.30
RAB9A P51151 2/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
G6PD P11413 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699664 0.86 MMP1 (0.41) ERBB2NQO2
SCHEMBL9700956 0.83 TSHR (0.37) ERBB2NQO2MEN1KMT2AMAPT
SCHEMBL9700960 0.81 MAPT (0.35) ERBB2MEN1KMT2AMAPTKDM4E
SCHEMBL9740990 0.81 MAPT (0.35) ERBB2MEN1KMT2AMAPTKDM4E
SCHEMBL4177978 0.79 ERBB2 (0.61) ERBB2NQO2MEN1KMT2AMAPT
SCHEMBL9746062 0.76 MMP1 (0.36)
SCHEMBL9163760 0.73 TSHR (0.42) NQO2MEN1KMT2AMAPTKDM4E
SCHEMBL9701973 0.71 NQO2 (0.39) NQO2MAPTKDM4E
SCHEMBL8645097 0.71 KMT2A (0.36) MEN1KMT2AMAPTKDM4E
SCHEMBL8644084 0.71 KMT2A (0.36) ERBB2MEN1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992014740-A1 QUINOXALINE PHOSPHONO-AMINO ACIDS AMERICAN HOME PRODUCTS CORPORATION (US) 1992-09-03 WO disclosed
US-5118675-A Therapy for central nervous system disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-02 US disclosed