SCHEMBL9701706

SCHEMBL9701706

CCN(CC)CC1Cn2c(C)cc3cccc(c32)O1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.36
HPGD P15428 2/20 0.32
HSD17B10 Q99714 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HRH1 P35367 1/20 0.32
TSHR P16473 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GRM2 Q14416 1/20 0.30
USP2 O75604 1/20 0.30
MAPK1 P28482 1/20 0.30
RAB9A P51151 1/20 0.30
TP53 P04637 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700002 0.81 HPGD (0.34) SLC6A4HPGDHSD17B10KDM4EALDH1A1
SCHEMBL9700179 0.77 ADRA2A (0.43) TSHRUSP2
SCHEMBL9699368 0.75 HRH3 (0.46) HTR2AHTR2CHRH1TSHRUSP2
SCHEMBL9700364 0.74 ADRA2A (0.35) TSHRUSP2
SCHEMBL9700471 0.71 CNR2 (0.35) SLC6A4ALDH1A1HTR2AHTR2CTSHR
SCHEMBL9699225 0.69 HTR2A (0.42) HPGDNISCHHTR2AHTR2CHRH1
SCHEMBL9700296 0.66 HTR2A (0.40) HPGDNISCHHTR2AHTR2CHRH1
SCHEMBL18258200 0.62 MCL1 (0.48) HTR2AHTR2C
SCHEMBL3785969 0.62 HTR1A (0.41) SLC6A4HPGDKDM4ENISCH
SCHEMBL3404272 0.62 HTR1A (0.41) SLC6A4HPGDKDM4ENISCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed