SCHEMBL9700296

SCHEMBL9700296

CCN(CC)CC1CN(N=O)c2ccccc2O1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HRH1 P35367 1/20 0.40
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TP53 P04637 4/20 0.38
THRB P10828 3/20 0.38
MAPT P10636 2/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
CA2 P00918 1/20 0.36
LTA4H P09960 1/20 0.35
NISCH Q9Y2I1 1/20 0.34
P2RX4 Q99571 1/20 0.34
ALOX5 P09917 1/20 0.34
HPGD P15428 1/20 0.34
GAA P10253 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699225 0.79 HTR2A (0.42) HTR2AHTR2CHRH1LMNASMN1; SMN2
SCHEMBL9701639 0.79 HTR1A (0.37) TP53THRBMAPTCA2ALOX5
SCHEMBL9153909 0.79 THRB (0.39) TP53THRBMAPTMEN1KMT2A
SCHEMBL9701358 0.78 HTR6 (0.41) HTR2AHTR2CHRH1LMNATP53
SCHEMBL9153937 0.76 HTT (0.38) TP53THRBMAPTMEN1KMT2A
SCHEMBL9154311 0.75 HTT (0.43) LMNASMN1; SMN2TP53THRBMAPT
SCHEMBL9700419 0.74 ADRA2A (0.56) HTR2AHTR2CHRH1
SCHEMBL9700016 0.74 ADRA2A (0.52)
SCHEMBL9700515 0.74 HRH3 (0.47) HTR2A
SCHEMBL30453493 0.73 MEN1 (0.44) LMNATP53THRBMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed