SCHEMBL9702570

SCHEMBL9702570

COc1ccc(CC2CNc3c(cc(Br)cc3[N+](=O)[O-])CN2)cc1OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.42
MAPK1 P28482 3/20 0.42
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4D Q08499 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
TNF P01375 1/20 0.42
LMNA P02545 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
NFKB1 P19838 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP2C19 P33261 1/20 0.39
TTR P02766 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11556653 0.68 PDE4A (0.77) MAPTMAPK1PDE4APDE4BPDE4D
SCHEMBL11157701 0.68 LMNA (0.47) MAPK1LMNAKDM4EALDH1A1
Hydrochloric Acid SCHEMBL11150663 0.67 LMNA (0.46) MAPK1LMNAKDM4EALDH1A1
SCHEMBL9852941 0.65 SMN1; SMN2 (0.46) CYP1A2LMNACYP2C19ALDH1A1HTT
SCHEMBL7351948 0.63 DRD2 (0.33) MAPTKDM4EALDH1A1
SCHEMBL7344244 0.63 AKR1B1 (0.38) MAPTCYP3A4ALDH1A1
SCHEMBL7346523 0.63 AKR1B1 (0.36) MAPTKMT2AALDH1A1HTT
SCHEMBL16181522 0.63 CYP1A2 (0.60) MAPTMAPK1CYP1A2CYP3A4KDM4E
Hydrochloric Acid SCHEMBL7343407 0.62 AKR1B1 (0.37) MAPTCYP3A4ALDH1A1
SCHEMBL16831402 0.62 MAPK1 (0.43) MAPTMAPK1CYP3A4LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992013860-A1 NEW 4,5,6,7-TETRAHYDRO-IMIDAZO-[4,5,lJK][1,4]-BENZODIAZEPINE-2-(1H)-THIONES, A METHOD OF PREPARING THEM AS WELL AS DRUGS CONTAINING THEM, AND INTERMEDIATES FOR THE PREPARATION OF THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1992-08-20 WO disclosed