SCHEMBL9703791

SCHEMBL9703791

CC(CC(=O)O)Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.53
MMP8 P22894 1/20 0.49
MMP14 P50281 1/20 0.49
CA14 Q9ULX7 1/20 0.49
EPHX1 P07099 1/20 0.47
EPHX2 P34913 1/20 0.47
ALDH1A1 P00352 2/20 0.46
APEX1 P27695 1/20 0.45
FFAR1 O14842 1/20 0.44
FNTA P49354 1/20 0.44
FNTB P49356 1/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA5A P35218 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703108 0.86 TSHR (0.59) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL5860319 0.81 MEN1 (0.47) CYP3A4ALDH1A1FFAR1FNTAFNTB
SCHEMBL5860329 0.81 MEN1 (0.47) CYP3A4ALDH1A1FFAR1FNTAFNTB
SCHEMBL13664802 0.80 MEN1 (0.50) ALDH1A1RAB9AMEN1KMT2ACA2
SCHEMBL735232 0.80 MMP8 (0.50) CYP3A4MMP8MMP14CA14EPHX1
SCHEMBL10914038 0.79 HPGD (0.55) ALDH1A1NPC1RAB9AMEN1KMT2A
SCHEMBL1823678 0.79 ALDH1A1 (0.45) CYP3A4MMP8MMP14CA14EPHX1
SCHEMBL1823681 0.79 ALDH1A1 (0.45) CYP3A4MMP8MMP14CA14EPHX1
SCHEMBL1555336 0.78 MMP8 (0.53) CYP3A4MMP8MMP14CA14EPHX1
SCHEMBL733499 0.78 MMP8 (0.53) CYP3A4MMP8MMP14CA14EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009119528-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2009-10-01 WO disclosed
EP-0203795-B1 Benzo [i,j] quinolizine-2-carboxylic acid derivatives, the salts and their hydrates, pharmaceutical compositions thereof, and process for preparing the same TOKYO TANABE COMPANY LIMITED (JP) 1992-07-29 EP disclosed
US-4720495-A Benzo[ij]quinolizine-2-carboxylic acids useful for treating bacterial infection TOKYO TANABE CO. LIMITED (JP) 1988-01-19 US disclosed
EP-0203795-A2 Benzo [i,j] quinolizine-2-carboxylic acid derivatives, the salts and their hydrates, pharmaceutical compositions thereof, and process for preparing the same TOKYO TANABE COMPANY LIMITED (JP) 1986-12-03 EP disclosed