SCHEMBL9704494

SCHEMBL9704494

COc1cc(S(C)(=O)=O)ccc1-c1nc2cc3c(cc2[nH]1)n(C)c(=O)c(=O)n3C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.47
CCNA2 P20248 1/20 0.47
CCND1 P24385 1/20 0.47
CDK2 P24941 1/20 0.47
CCND3 P30281 1/20 0.47
NPBWR1 P48145 1/20 0.42
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
SCD O00767 5/20 0.41
AMY1A P0DUB6 1/20 0.41
CBFB Q13951 1/20 0.39
FADS1 O60427 1/20 0.39
PDE5A O76074 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
BRPF1 P55201 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10552928 0.88 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9703335 0.82 CDK4 (0.47) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9705442 0.82 KDM4E (0.41) KDM4ECYP1A2CYP3A4AMY1APDE5A
SCHEMBL9702805 0.80 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9703323 0.79 CDK4 (0.47) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10853376 0.79 CDK4 (0.46) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10552771 0.78 KDM4E (0.40) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10765238 0.78 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10677421 0.78 PDE5A (0.50) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9702854 0.76 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed