SCHEMBL9702805

SCHEMBL9702805

COc1cc(S(C)(=O)=O)ccc1-c1nc2cc3[nH]c(=O)cnc3cc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.45
CCNA2 P20248 1/20 0.45
CCND1 P24385 1/20 0.45
CDK2 P24941 1/20 0.45
CCND3 P30281 1/20 0.45
NPBWR1 P48145 1/20 0.43
CBFB Q13951 1/20 0.42
SCD O00767 7/20 0.41
AMY1A P0DUB6 1/20 0.41
PDE5A O76074 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
ATR Q13535 1/20 0.41
FADS1 O60427 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703335 0.85 CDK4 (0.47) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10853376 0.82 CDK4 (0.46) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9702924 0.82 AMY1A (0.41) AMY1APDE5APDE3BPDE3A
SCHEMBL10677421 0.81 PDE5A (0.50) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9704494 0.80 CDK4 (0.47) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL9702854 0.79 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10765238 0.79 CDK4 (0.45) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL7272031 0.79 PDE5A (0.54) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL11021893 0.78 ATR (0.44) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL11021898 0.78 ATR (0.53) CDK4CCNA2CCND1CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed
EP-0275888-A2 Tricyclic benzimidazoles, process for their preparation and use as medicaments Roche Diagnostics GmbH (DE) 1988-07-27 EP disclosed