SCHEMBL9705442

SCHEMBL9705442

COc1cc([S+](C)[O-])ccc1-c1nc2cc3c(cc2[nH]1)n(C)c(=O)c(=O)n3C

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
AMY1A P0DUB6 12/20 0.40
PDE5A O76074 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
ADORA2B P29275 1/20 0.36
PDE2A O00408 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10551908 0.88 AMY1A (0.39) KDM4ECYP1A2CYP3A4AMY1APDE5A
SCHEMBL9703649 0.83 AMY1A (0.43) AMY1APDE5APDE3BPDE3APDE2A
SCHEMBL9704494 0.82 CDK4 (0.47) KDM4ECYP1A2CYP3A4AMY1APDE5A
SCHEMBL9702924 0.80 AMY1A (0.41) KDM4ECYP1A2AMY1APDE5APDE3B
SCHEMBL10852513 0.80 AMY1A (0.40) KDM4ECYP1A2AMY1APDE5APDE3B
SCHEMBL9704539 0.79 AMY1A (0.40) AMY1APDE5APDE3BPDE3A
SCHEMBL10373752 0.78 PDE3B (0.48) KDM4ECYP1A2AMY1APDE5APDE3B
SCHEMBL9704436 0.77 PDE5A (0.43) KDM4ECYP1A2AMY1APDE5APDE3B
SCHEMBL9703428 0.77 PDE3B (0.41) KDM4ECYP1A2AMY1APDE5APDE3B
SCHEMBL10742305 0.77 PDE5A (0.47) KDM4ECYP1A2AMY1APDE5APDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed