SCHEMBL9704732

SCHEMBL9704732

CCCCc1nc2nc(NC3CCCCC3)ncc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 1/20 0.53
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
CCND2 P30279 1/20 0.41
CCND3 P30281 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
LMNA P02545 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
FLT3 P36888 4/20 0.39
TYRO3 Q06418 4/20 0.39
MERTK Q12866 4/20 0.39
GAS6 Q14393 4/20 0.39
CDK2 P24941 2/20 0.38
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
AXL P30530 1/20 0.37
POLA1 P09884 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704728 0.82 PDE4A (0.43) PAK1CDK4CCND1CCND2CCND3
SCHEMBL9704936 0.77 POLA1 (0.41) FLT3TYRO3MERTKGAS6AXL
SCHEMBL9705994 0.72 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL15264150 0.70 PAK1 (1.00) PAK1LMNAADORA3CDK2CDK1
SCHEMBL9705260 0.69 NOS1 (0.45)
SCHEMBL9706008 0.69 NOS3 (0.40)
SCHEMBL15545184 0.68 PAK1 (0.97) PAK1LMNAADORA3CDK2POLA1
SCHEMBL18786068 0.67 PI4KA (0.44)
SCHEMBL7851163 0.67 PI4KA (0.49)
SCHEMBL30523392 0.66 PAK1 (0.91) PAK1LMNAADORA3CDK2POLA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470543-A1 Heterocyclic imidazoles, remedies containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-02-12 EP disclosed