SCHEMBL9704866

SCHEMBL9704866

CC(=O)N(c1ccc(O)cc1)c1ccc2cc(O)ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 8/20 0.49
ESR2 Q92731 8/20 0.49
CYP1A2 P05177 1/20 0.41
ESRRG P62508 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CLK1 P49759 2/20 0.39
DYRK1A Q13627 2/20 0.39
DYRK1B Q9Y463 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HSD17B10 Q99714 2/20 0.38
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38
HIF1A Q16665 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703005 0.85 MEN1 (0.46) ESR1ESR2CYP1A2NPC1RAB9A
SCHEMBL7153902 0.84 ESR1 (0.47) ESR1ESR2NPC1RAB9AMEN1
SCHEMBL25969111 0.81 CYP1A2 (0.43) ESR1ESR2CYP1A2ESRRGNPC1
SCHEMBL1176872 0.79 ESR1 (0.49) ESR1ESR2CYP1A2NPC1RAB9A
SCHEMBL3975700 0.77 NPSR1 (0.52) ESR1ESR2NPC1RAB9AMEN1
SCHEMBL2038478 0.76 ESR1 (0.46) ESR1ESR2CYP1A2NPC1RAB9A
SCHEMBL25969113 0.76 ESR1 (0.42) ESR1ESR2CYP1A2NPC1RAB9A
SCHEMBL712464 0.75 ESR1 (0.42) ESR1ESR2CYP1A2ESRRGNPC1
SCHEMBL28269013 0.72 TSHR (0.56) ESR1ESR2CYP1A2NPC1MEN1
SCHEMBL1680160 0.72 CYP1A2 (0.54) ESR1ESR2CYP1A2HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0221677-B1 P-AMINOPHENOLS, DERIVATIVES THEREOF AND USE FOR MANUFACTURE OF A MEDICAMENT E.R. Squibb & Sons, Inc. (US) 1992-09-09 EP disclosed
US-4910208-A Skin disorders, antiinflammatory agent E. R. SQUIBB & SONS, INC. (US) 1990-03-20 US disclosed
US-4814454-A ANTIALLERGENS, ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1989-03-21 US disclosed
EP-0221677-A2 p-Aminophenols, derivatives thereof and use for manufacture of a medicament E.R. Squibb & Sons, Inc. (US) 1987-05-13 EP disclosed