SCHEMBL9705738

SCHEMBL9705738

COC(=O)c1cc(Cl)c(OCCCCCc2cc(C)no2)c(Br)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
CYP2D6 P10635 3/20 0.41
CYP1A2 P05177 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
CYP3A4 P08684 2/20 0.38
NR1I2 O75469 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC6 Q9UBN7 3/20 0.38
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
KLK1 P06870 1/20 0.36
THRA P10827 2/20 0.35
THRB P10828 2/20 0.35
POLB P06746 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9705669 0.93 CYP2D6 (0.41) KDM4ECYP2D6CYP1A2ALDH1A1TDP1
SCHEMBL9706270 0.90 KDM4E (0.42) KDM4ECYP2D6CYP1A2ALDH1A1TDP1
SCHEMBL9706267 0.86 KDM4E (0.41) KDM4ECYP2D6CYP1A2ALDH1A1TDP1
SCHEMBL9705709 0.84 MAPT (0.40) KDM4ECYP2D6ALDH1A1MEN1KMT2A
SCHEMBL9200429 0.82 PLAU (0.49) KDM4ECYP2D6MEN1KMT2ACYP3A4
SCHEMBL9436198 0.81 LMNA (0.42) KDM4ECYP2D6ALDH1A1MEN1KMT2A
SCHEMBL9862957 0.79 CYP3A4 (0.44) KDM4ECYP2D6TDP1CYP3A4NR1I2
SCHEMBL8875953 0.79 NR1I2 (0.55) CYP2D6ALDH1A1MEN1KMT2ACYP3A4
SCHEMBL9706268 0.79 NR1I2 (0.45) KDM4ECYP2D6ALDH1A1TDP1CYP3A4
SCHEMBL10413619 0.78 NR1I2 (0.44) KDM4ECYP2D6ALDH1A1TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0207454-B1 ISOXAZOLE AND FURAN DERIVATIVES, THEIR PREPARATION AND USE AS ANTIVIRAL AGENTS STERLING WINTHROP INC. (US) 1992-09-09 EP disclosed
US-5002960-A Viricides for combating picornaviruses STERLING DRUG, INC. (US) 1991-03-26 US disclosed
US-4939267-A Viricides STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4843087-A OXAZOLINYL COMPOUNDS; RHINOVIRUSES AND PICORNAVIRUSES STERLING DRUG INC. (US) 1989-06-27 US disclosed
EP-0207454-A2 Isoxazole and furan derivatives, their preparation and use as antiviral agents STERLING WINTHROP INC. (US) 1987-01-07 EP disclosed