SCHEMBL9706609

SCHEMBL9706609

CCn1c(=O)[nH]c(=S)c2[nH]c(C)nc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.49
HTT P42858 2/20 0.49
ADORA2A P29274 3/20 0.42
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
PDE2A O00408 1/20 0.41
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
PDE1C Q14123 1/20 0.41
SIRT1 Q96EB6 2/20 0.38
SIRT3 Q9NTG7 2/20 0.38
SIRT5 Q9NXA8 2/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
CYP1A2 P05177 3/20 0.35
LMNA P02545 2/20 0.35
CYP3A4 P08684 2/20 0.35
MAPK1 P28482 2/20 0.35
PMP22 Q01453 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9706669 0.88 ADORA2A (0.45) HPGDHTTADORA2APDE4APDE4B
SCHEMBL7419694 0.85 PDE4A (0.47) HPGDADORA2APDE4APDE4BPDE4C
SCHEMBL10963141 0.83 ADORA2A (0.55) HPGDHTTADORA2APDE4APDE4B
SCHEMBL1460912 0.83 PDE1A (0.58) HPGDHTTPDE2APDE1APDE1B
SCHEMBL9706596 0.83 ADORA2A (0.41) HPGDHTTADORA2APDE4APDE4B
SCHEMBL7423089 0.80 ADORA2A (0.39) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9645623 0.78 CYP3A4 (0.45) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7676923 0.78 ADORA1 (0.56) ADORA2ACYP1A2LMNAPMP22MEN1
SCHEMBL7863965 0.74 ADORA2B (0.58) HPGDADORA2ACYP1A2CYP3A4MAPK1
SCHEMBL28143495 0.73 SIRT1 (0.67) HPGDADORA2APDE2APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4820709-A 6-thioxanthine derivatives EUROCELTIQUE, S.A. (LU) 1989-04-11 US claimed
CN-86101050-A The manufacture method of 6-Thioxanthine derivatives and application thereof 1986-11-12 CN claimed
EP-0191313-B1 6-THIOXANTHINE DERIVATIVES Euro-Celtique S.A. (LU) 1992-10-28 EP disclosed
CN-1013676-B 6-THIOXANTHINE DERIVATIVES EURO CELTIQUE SA (US) 1991-08-28 CN disclosed
US-4820709-A 6-thioxanthine derivatives EUROCELTIQUE, S.A. (LU) 1989-04-11 US disclosed
US-4710503-A 6-thioxanthine derivatives EUROCELTIQUE S.A. (LU) 1987-12-01 US disclosed
CN-86101050-A The manufacture method of 6-Thioxanthine derivatives and application thereof 1986-11-12 CN disclosed
EP-0191313-A1 6-Thioxanthine derivatives Euro-Celtique S.A. (LU) 1986-08-20 EP disclosed