SCHEMBL9707085

SCHEMBL9707085

O=C(CCSc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1)N1CCCC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 11/20 0.68
RAB9A P51151 8/20 0.68
NPC1 O15118 8/20 0.68
ALDH1A1 P00352 8/20 0.68
HPGD P15428 3/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
USP2 O75604 1/20 0.53
MAPT P10636 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
NAAA Q02083 1/20 0.49
POLB P06746 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 2/20 0.45
TSHR P16473 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9510615 0.89 SMN1; SMN2 (0.53) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
SCHEMBL9814008 0.89 SMN1; SMN2 (0.70) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL9513854 0.88 SMN1; SMN2 (0.52) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
SCHEMBL9510247 0.86 SMN1; SMN2 (0.50) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
Hydrochloric Acid SCHEMBL9513665 0.85 SMN1; SMN2 (0.49) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
SCHEMBL9528422 0.81 SMN1; SMN2 (0.97) SMN1; SMN2RAB9ANPC1ALDH1A1HPGD
SCHEMBL9550710 0.81 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL9707052 0.80 ACE (0.46) SMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL9813051 0.78 PTPN1 (0.44) SMN1; SMN2RAB9ANPC1ALDH1A1CYP1A2
SCHEMBL9814016 0.78 SMN1; SMN2 (0.49) SMN1; SMN2RAB9ANPC1ALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0190685-B1 HETEROCYCLIC AMIDES G.D. Searle & Co. (US) 1992-07-01 EP disclosed
US-4981853-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS G. D. SEARLE & CO. (US) 1991-01-01 US disclosed
US-4959364-A Method of treating inflammation, allergy, asthma and proliferative skin disease using heterocyclic amides G. D. SEARLE & CO. (US) 1990-09-25 US disclosed
EP-0190685-A2 Heterocyclic amides G.D. Searle & Co. (US) 1986-08-13 EP disclosed