SCHEMBL9707052

SCHEMBL9707052

O=C(O)[C@@H]1CCCN1C(=O)CCSc1cc(-c2ccccc2)c(O)c(-c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE P12821 15/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
ACE2 Q9BYF1 5/20 0.45
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9814010 0.89 ACE (0.49) ACENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9707078 0.82 ACE (0.49) ACECHRM2CHRM4CHRM1CHRM3
SCHEMBL9707085 0.80 SMN1; SMN2 (0.68) NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9707098 0.79 ACE (0.43) ACECHRM2CHRM4CHRM1CHRM3
SCHEMBL11547220 0.77 NPC1 (0.59) ACECHRM2CHRM4CHRM1CHRM3
SCHEMBL11548414 0.76 ACE (0.52) ACECHRM2CHRM4CHRM1CHRM3
SCHEMBL9510615 0.75 SMN1; SMN2 (0.53) NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL9814008 0.75 SMN1; SMN2 (0.70) NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL11544959 0.74 DPP4 (0.49) ACECHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL9513854 0.74 SMN1; SMN2 (0.52) NPC1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0190685-B1 HETEROCYCLIC AMIDES G.D. Searle & Co. (US) 1992-07-01 EP disclosed
US-4981853-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS G. D. SEARLE & CO. (US) 1991-01-01 US disclosed
US-4959364-A Method of treating inflammation, allergy, asthma and proliferative skin disease using heterocyclic amides G. D. SEARLE & CO. (US) 1990-09-25 US disclosed
EP-0190685-A2 Heterocyclic amides G.D. Searle & Co. (US) 1986-08-13 EP disclosed