SCHEMBL9707562

SCHEMBL9707562

COC(=O)Cn1c(=O)n(CC(C)C)c(=O)c2c1nc(C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.39
AGTR2 P50052 2/20 0.39
KMT2A Q03164 2/20 0.39
ADORA3 P0DMS8 4/20 0.39
ADORA1 P30542 2/20 0.39
PPARG P37231 4/20 0.38
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707646 0.97 KMT2A (0.41) AGTR1AGTR2KMT2AADORA3ADORA1
SCHEMBL9708749 0.94 KMT2A (0.44) AGTR1AGTR2KMT2AADORA3PPARG
SCHEMBL9708195 0.92 PPARG (0.39) AGTR1AGTR2KMT2AADORA3ADORA1
SCHEMBL9707465 0.92 KMT2A (0.44) AGTR1AGTR2KMT2AADORA3PPARG
SCHEMBL9707686 0.91 AGTR1 (0.43) AGTR1AGTR2KMT2AADORA3ADORA1
SCHEMBL9707851 0.90 AGTR1 (0.43) AGTR1AGTR2KMT2AADORA3ADORA1
SCHEMBL9707687 0.90 AGTR1 (0.46) AGTR1AGTR2PPARG
SCHEMBL9707859 0.90 DCTPP1 (0.40) AGTR1AGTR2KMT2AADORA3PPARG
SCHEMBL9707855 0.90 AGTR1 (0.39) AGTR1AGTR2KMT2APPARG
SCHEMBL9707476 0.89 TSHR (0.41) AGTR1AGTR2KMT2APPARGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed