SCHEMBL9708058

SCHEMBL9708058

CCCn1c(=O)n(CCOC)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 13/20 0.40
ADORA1 P30542 4/20 0.40
ADORA2A P29274 4/20 0.38
ADORA2B P29275 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708153 1.00 ADORA3 (0.40) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9708263 0.95 ADORA3 (0.39) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9708050 0.95 ADORA2A (0.39) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9707535 0.95 ADORA3 (0.43) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9708824 0.93 ADORA3 (0.41) ADORA3ADORA2AADORA2B
SCHEMBL9708259 0.93 ADORA3 (0.41) ADORA3ADORA2AADORA2B
SCHEMBL9708628 0.92 USP2 (0.41) ADORA3ADORA2AADORA2B
SCHEMBL9707714 0.92 DCTPP1 (0.44) ADORA2AADORA2B
SCHEMBL9708213 0.92 ADORA3 (0.42) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL9708283 0.92 ADORA3 (0.41) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed