SCHEMBL9708824

SCHEMBL9708824

COCCn1c(=O)n(CCc2ccccc2)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.41
ADORA2B P29275 3/20 0.40
ADORA2A P29274 1/20 0.40
AGTR1 P30556 5/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DCTPP1 Q9H773 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AGTR2 P50052 1/20 0.37
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708259 1.00 ADORA3 (0.41) ADORA3ADORA2BADORA2AAGTR1ALDH1A1
SCHEMBL9707877 0.95 AGTR1 (0.42) ADORA3AGTR1ALDH1A1MEN1KMT2A
SCHEMBL9708263 0.93 ADORA3 (0.39) ADORA3ADORA2BADORA2AAGTR1ALDH1A1
SCHEMBL9708153 0.93 ADORA3 (0.40) ADORA3ADORA2BADORA2A
SCHEMBL9708058 0.93 ADORA3 (0.40) ADORA3ADORA2BADORA2A
SCHEMBL9708050 0.92 ADORA2A (0.39) ADORA3ADORA2BADORA2AAGTR1ALDH1A1
SCHEMBL9707297 0.92 ADORA3 (0.43) ADORA3ADORA2BADORA2AAGTR1AGTR2
SCHEMBL9707529 0.92 ADORA3 (0.43) ADORA3ADORA2BADORA2AAGTR1AGTR2
SCHEMBL9708598 0.92 ADORA1 (0.44) ADORA3ADORA2BADORA2AAGTR1TSHR
SCHEMBL9708045 0.91 ADORA3 (0.42) ADORA3ADORA2BADORA2AAGTR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed