SCHEMBL9708299

SCHEMBL9708299

CCc1nc2c(c(=O)[nH]c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
TPH1 P17752 1/20 0.48
TPH2 Q8IWU9 1/20 0.48
RAB9A P51151 2/20 0.47
USP2 O75604 1/20 0.47
POLB P06746 2/20 0.47
BRAF P15056 1/20 0.47
AGTR1 P30556 1/20 0.47
AGTR2 P50052 1/20 0.47
TP53 P04637 1/20 0.46
ALDH1A1 P00352 2/20 0.46
CXCL8 P10145 2/20 0.46
NOD2 Q9HC29 2/20 0.46
NOD1 Q9Y239 2/20 0.46
KDM4E B2RXH2 1/20 0.46
TNF P01375 1/20 0.46
MAPT P10636 1/20 0.46
G6PD P11413 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708629 0.93 AGTR1 (0.48) MEN1KMT2ATPH1TPH2RAB9A
SCHEMBL9707992 0.91 USP2 (0.51) MEN1KMT2ARAB9AUSP2AGTR1
SCHEMBL9708861 0.91 TPH1 (0.51) MEN1KMT2ATPH1TPH2RAB9A
SCHEMBL9708297 0.91 MEN1 (0.54) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707996 0.91 USP2 (0.52) MEN1KMT2ATPH1TPH2RAB9A
SCHEMBL9708307 0.91 MEN1 (0.47) MEN1KMT2ATPH1TPH2RAB9A
SCHEMBL9708384 0.90 MEN1 (0.48) MEN1KMT2ATPH1TPH2USP2
SCHEMBL9708366 0.89 BRAF (0.48) MEN1KMT2ARAB9APOLBBRAF
SCHEMBL9708587 0.89 AGTR1 (0.45) MEN1KMT2ATPH1TPH2AGTR1
SCHEMBL9707846 0.88 ALDH1A1 (0.49) MEN1KMT2ATPH1TPH2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed