SCHEMBL9708337

SCHEMBL9708337

CCCn1c(=O)c2c(nc(CC)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(C)c1=O

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 5/20 0.44
AGTR2 P50052 5/20 0.44
ALOX15 P16050 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA1 P30542 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708359 0.95 AGTR1 (0.45) AGTR1AGTR2ADORA3ADORA1
SCHEMBL9708536 0.94 AGTR1 (0.46) AGTR1AGTR2ALOX15HSD17B10MAPT
SCHEMBL9708840 0.94 AGTR1 (0.44) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707817 0.93 AGTR1 (0.44) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9708275 0.93 TSHR (0.46) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9707515 0.93 AGTR1 (0.50) AGTR1AGTR2
SCHEMBL9708324 0.92 ADORA3 (0.43) AGTR1AGTR2ADORA3ADORA1
SCHEMBL9707699 0.92 ALOX15 (0.52) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9708878 0.92 ALOX15 (0.41) AGTR1AGTR2ALOX15HSD17B10ALDH1A1
SCHEMBL9708070 0.92 AGTR1 (0.48) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed