SCHEMBL9708401

SCHEMBL9708401

COCCn1c(=O)c2c(nc(CC(C)(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CC2CC2)c1=O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 8/20 0.42
PDE4A P27815 8/20 0.42
PDE4B Q07343 8/20 0.42
PDE4C Q08493 8/20 0.42
PDE4D Q08499 8/20 0.42
ADORA3 P0DMS8 8/20 0.37
AGTR1 P30556 1/20 0.37
AGTR2 P50052 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ADORA2A P29274 2/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
ADORA2B P29275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707595 0.93 PDE5A (0.47) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9708546 0.92 PDE5A (0.42) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9708807 0.92 PDE5A (0.43) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9707532 0.91 AGTR1 (0.42) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9708153 0.91 ADORA3 (0.40) ADORA3ADORA2AADORA2B
SCHEMBL9708263 0.91 ADORA3 (0.39) ADORA3AGTR1AGTR2ADORA2AADORA2B
SCHEMBL9708058 0.91 ADORA3 (0.40) ADORA3ADORA2AADORA2B
SCHEMBL9708627 0.91 PDE5A (0.43) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9707536 0.90 PDE5A (0.43) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9708893 0.90 PDE5A (0.44) PDE5APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed