SCHEMBL9708734

SCHEMBL9708734

CCCn1c(=O)n(C)c(=O)c2c1nc(CC(C)(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.39
AGTR1 P30556 2/20 0.39
AGTR2 P50052 2/20 0.39
HPGD P15428 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707535 0.95 ADORA3 (0.43) AGTR1AGTR2ADORA3
SCHEMBL9707475 0.94 ALOX15 (0.41) ALOX15HSD17B10HTTNPSR1ALDH1A1
SCHEMBL9708004 0.94 ADORA3 (0.40) AGTR1AGTR2ADORA3
SCHEMBL9708878 0.94 ALOX15 (0.41) ALOX15HSD17B10HTTNPSR1ALDH1A1
SCHEMBL9708283 0.93 ADORA3 (0.41) AGTR1AGTR2ADORA3
SCHEMBL9707632 0.92 ALOX15 (0.43) ALOX15HSD17B10HTTNPSR1ALDH1A1
SCHEMBL9707817 0.92 AGTR1 (0.44) ALOX15HSD17B10HTTNPSR1ALDH1A1
SCHEMBL9708628 0.91 USP2 (0.41) ALOX15HSD17B10HTTNPSR1ALDH1A1
SCHEMBL9707374 0.91 AGTR1 (0.46) ALOX15HSD17B10AGTR1AGTR2
SCHEMBL9708090 0.91 ADORA3 (0.39) AGTR1AGTR2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed