SCHEMBL9709146

SCHEMBL9709146

NC(=O)C(NC(=O)CCc1ccccc1)C1NCCS1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CYP1A2 P05177 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HDAC1 Q13547 3/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
MMP2 P08253 1/20 0.39
MMP8 P22894 1/20 0.39
MMP12 P39900 1/20 0.39
MMP13 P45452 1/20 0.39
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP2C19 P33261 1/20 0.38
CNR2 P34972 1/20 0.37
ITGB3 P05106 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709176 0.77 CNR2 (0.43) CYP1A2MMP2HPGDALDH1A1CYP2C19
SCHEMBL9709042 0.74 CYP1A2 (0.46) CYP1A2ALDH1A1
SCHEMBL9604373 0.74 NPY1R (0.42) HDAC2HDAC8HDAC6CYP1A2NPC1
SCHEMBL1903649 0.69 HDAC2 (0.54) HDAC2HDAC8HDAC6RAB9AHDAC1
SCHEMBL21587872 0.69 HDAC2 (0.54) HDAC2HDAC8HDAC6RAB9AHDAC1
SCHEMBL24533878 0.67 MMP2 (0.58) HDAC2HDAC8HDAC6HDAC1MAPT
SCHEMBL24533867 0.67 MMP2 (0.58) HDAC2HDAC8HDAC6HDAC1MAPT
SCHEMBL16359253 0.67 HDAC2 (0.53) HDAC2HDAC8HDAC6HDAC1MAPT
SCHEMBL9708917 0.67 CNR2 (0.40) CYP1A2ALDH1A1CYP2C19CNR2
SCHEMBL16908006 0.66 HDAC2 (0.51) HDAC2HDAC8HDAC6RAB9AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992020665-A1 THIAZOLIDINE DERIVATIVES AND THEIR USE IN THERAPY GLAXO GROUP LIMITED (GB) 1992-11-26 WO disclosed