SCHEMBL9709749

SCHEMBL9709749

Cc1cc(NCc2ccc(-c3ccccc3C(=O)O)cc2)c2cccc(C)c2n1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CD38 P28907 14/20 0.64
CYP3A4 P08684 4/20 0.55
KCNH2 Q12809 1/20 0.55
BDKRB1 P46663 1/20 0.48
PPARG P37231 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3051435 0.88 CD38 (0.60) CD38CYP3A4KCNH2
SCHEMBL3058636 0.87 CD38 (0.56) CD38BDKRB1
Hydrochloric Acid SCHEMBL9494706 0.86 CD38 (0.55) CD38BDKRB1
SCHEMBL9363742 0.82 CD38 (0.69) CD38CYP3A4KCNH2
SCHEMBL9709700 0.82 VCP (0.52) CD38BDKRB1PPARG
SCHEMBL9709814 0.79 CD38 (0.55) CD38BDKRB1PPARG
SCHEMBL9709608 0.79 CD38 (0.50) CD38BDKRB1
SCHEMBL9709799 0.79 CD38 (0.47) CD38BDKRB1PPARG
SCHEMBL9494718 0.78 ACP1 (0.54) CD38BDKRB1
SCHEMBL20680363 0.78 CD38 (1.00) CD38CYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO claimed
WO-1992022533-A1 4-AMINOQUINOLINES AND PHARMACEUTICAL COMPOSITIONS THEREOF THE UPJOHN COMPANY (US) 1992-12-23 WO disclosed