SCHEMBL9709753

SCHEMBL9709753

CCCCC(=O)CCc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 6/20 0.42
IAPP P10997 1/20 0.42
AGTR1 P30556 9/20 0.42
ABCB11 O95342 1/20 0.39
GP6 Q9HCN6 1/20 0.39
BRS3 P32247 2/20 0.39
AGTR2 P50052 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9709732 0.97 LTB4R2 (0.41) LTB4R2IAPPAGTR1BRS3AGTR2
SCHEMBL9709552 0.93 IAPP (0.40) LTB4R2IAPPAGTR1BRS3AGTR2
SCHEMBL9709582 0.90 IAPP (0.39) LTB4R2IAPPAGTR1
SCHEMBL6953051 0.85 HSD11B1 (0.47) AGTR1BRS3AGTR2
SCHEMBL6957300 0.83 HSD11B1 (0.47) AGTR1AGTR2
SCHEMBL6949197 0.83 HSD11B1 (0.47) AGTR1AGTR2
SCHEMBL6961100 0.83 NPC1 (0.39) AGTR1AGTR2
SCHEMBL4609709 0.82 LTB4R2 (0.60) LTB4R2
SCHEMBL8524519 0.81 HSD11B1 (0.43) AGTR1
SCHEMBL8260354 0.81 LTB4R2 (0.52) LTB4R2AGTR1ABCB11GP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5157040-A Treatment of hypertension, ocular hypertension and some CNS disorders MERCK & CO., INC. (US) 1992-10-20 US disclosed
EP-0507594-A1 Substituted quinolines as angiotensin II antagonists MERCK & CO. INC. (US) 1992-10-07 EP disclosed