SCHEMBL9710299

SCHEMBL9710299

O=C1CSc2ccc(F)cc2CN1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
CHEK2 O96017 1/20 0.40
CDK1 P06493 1/20 0.40
PIM1 P11309 1/20 0.40
FGFR1 P11362 1/20 0.40
CDK2 P24941 1/20 0.40
MARK3 P27448 1/20 0.40
CSNK2A1 P68400 1/20 0.40
MARK2 Q7KZI7 1/20 0.40
NOTUM Q6P988 1/20 0.38
HTT P42858 2/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
ALDH1A1 P00352 2/20 0.36
EPHX2 P34913 1/20 0.36
PARP1 P09874 1/20 0.36
PARP10 Q53GL7 1/20 0.36
GRM5 P41594 2/20 0.35
SRD5A1 P18405 1/20 0.35
HSD17B3 P37058 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9710025 0.87 PARP1 (0.39) AURKACHEK2CDK1PIM1FGFR1
SCHEMBL8120667 0.76 MAOA (0.57) HTTMAOAMAOBLMNA
SCHEMBL8526616 0.75 RYR2 (0.47) MAOAMAOBALDH1A1EPHX2HSD17B3
SCHEMBL10509516 0.72 HTT (0.59) HTTMAOAMAOBALDH1A1EPHX2
SCHEMBL31441353 0.72 PARP1 (0.43) PARP1PARP10GRM5SRD5A1OPRM1
SCHEMBL31254528 0.72 PARP1 (0.43) PARP1PARP10GRM5SRD5A1OPRM1
SCHEMBL5751107 0.70 MAOB (0.64) HTTMAOAMAOBALDH1A1EPHX2
SCHEMBL5191132 0.70 PARP1 (0.39) MAOBPARP1PARP10GRM5SRD5A1
SCHEMBL29673299 0.70 CMA1 (0.45) HTTMAOAMAOBEPHX2PARP1
SCHEMBL31441323 0.69 PARP1 (0.41) PARP1PARP10GRM5SRD5A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021668-A1 BENZOTHIAZEPINONES AND THEIR USE AS ANTICONVULSANTS THE BOOTS COMPANY PLC (GB) 1992-12-10 WO claimed
WO-1992021668-A1 BENZOTHIAZEPINONES AND THEIR USE AS ANTICONVULSANTS THE BOOTS COMPANY PLC (GB) 1992-12-10 WO disclosed