SCHEMBL9713434

SCHEMBL9713434

Cc1ccc(C#Cc2ccc(OC(F)(F)F)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.40
ACACB O00763 4/20 0.40
ADRB3 P13945 1/20 0.39
TSPO P30536 1/20 0.39
KCNH2 Q12809 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
GPR35 Q9HC97 1/20 0.39
MCHR1 Q99705 2/20 0.38
RXRA P19793 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
GPR3 P46089 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713235 0.87 GRM5 (0.37) GRM5ACACBMCHR1
SCHEMBL9713366 0.85 ACACB (0.49) GRM5ACACBADRB3TSPOKCNH2
SCHEMBL9713010 0.83 ACACB (0.49) ACACBMCHR1RXRAGRIN1GRIN2B
SCHEMBL9816286 0.83 ACACB (0.52) ACACBMCHR1
SCHEMBL17225200 0.82 ACACB (0.48) GRM5ACACBKCNH2MCHR1GPR3
SCHEMBL9713133 0.82 RXRA (0.41) GRM5ACACBADRB3TSPOKCNH2
SCHEMBL4147154 0.81 MCHR1 (0.53) GRM5ACACBKCNH2MCHR1
SCHEMBL9713293 0.81 ACACB (0.51) ACACBMCHR1KMT2A
SCHEMBL9712769 0.81 ACACB (0.56) ACACBMCHR1
SCHEMBL14129682 0.81 GRM5 (0.53) GRM5ACACBKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164114-A LIQUID CRYSTAL MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1992-11-17 US disclosed
EP-0306521-B1 ETHINE DERIVATIVES AS COMPOUNDS OF LIQUID CRYSTAL PHASES MERCK PATENT GmbH (DE) 1991-10-16 EP disclosed
EP-0306521-A1 ETHINE DERIVATIVES AS COMPOUNDS OF LIQUID CRYSTAL PHASES. MERCK PATENT GMBH (DE) 1989-03-15 EP disclosed
WO-1988007516-A1 ETHINE DERIVATIVES AS COMPOUNDS OF LIQUID CRYSTAL PHASES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed