SCHEMBL9713617

SCHEMBL9713617

CCCNc1ccc(S(=O)(=O)c2ccc(NC(C)=O)cc2)c(NC)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
PKM P14618 2/20 0.47
POLB P06746 2/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 5/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
TP53 P04637 1/20 0.42
ATM Q13315 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714074 0.84 CA1 (0.44) GAAPKMCYP2C19CA1CA2
SCHEMBL9714041 0.75 ALDH1A1 (0.56) GAAPKMPOLBCYP2C19KMT2A
SCHEMBL8483061 0.74 SMN1; SMN2 (0.57) POLBCYP2C19KMT2AALDH1A1MAPT
SCHEMBL9713594 0.74 GAA (0.49) GAAPKMPOLBCYP2C19KMT2A
SCHEMBL9713778 0.71 CDK1 (0.68) GAAPKMPOLBCYP2C19KMT2A
SCHEMBL19392261 0.71 PKM (0.74) GAAPKMPOLBCYP2C19KMT2A
Acedapsone SCHEMBL152710 0.71 PKM (0.85) GAAPKMPOLBCYP2C19KMT2A
Acedapsone SCHEMBL22518385 0.69 PKM (0.82) GAAPKMPOLBCYP2C19KMT2A
Acedapsone SCHEMBL28716352 0.69 PKM (0.82) GAAPKMPOLBCYP2C19KMT2A
SCHEMBL9614881 0.69 POLB (0.84) GAAPOLBCYP2C19KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed