SCHEMBL9713778

SCHEMBL9713778

CCNc1ccc(S(=O)(=O)c2ccc(NC(C)=O)cc2)c(C(=O)OC)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.68
GAA P10253 1/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
HPGD P15428 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PKM P14618 2/20 0.47
TDP1 Q9NUW8 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 2/20 0.44
KMT2A Q03164 3/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
POLB P06746 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9713798 0.87 CDK1 (0.52) CDK1GAAALDH1A1KDM4EHPGD
SCHEMBL9713813 0.83 CDK1 (0.67) CDK1GAAALDH1A1KDM4EHPGD
SCHEMBL9714041 0.83 ALDH1A1 (0.56) GAAALDH1A1KDM4EHPGDPKM
SCHEMBL9713594 0.79 GAA (0.49) GAAALDH1A1PKMCYP2C19SMN1; SMN2
SCHEMBL9714037 0.74 PKM (0.46) CDK1GAAPKMTDP1CYP2C19
SCHEMBL9713905 0.74 PKM (0.46) GAAALDH1A1KDM4EHPGDPKM
SCHEMBL17477155 0.72 ALDH1A1 (0.72) CDK1ALDH1A1KDM4EHPGDCASP1
SCHEMBL21900515 0.72 KMT2A (0.58) GAAALDH1A1KDM4ETDP1SMN1; SMN2
SCHEMBL9713617 0.71 GAA (0.49) GAAALDH1A1KDM4EHPGDPKM
SCHEMBL9713853 0.71 PKM (0.67) CDK1GAAALDH1A1PKMCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed