SCHEMBL9713702

SCHEMBL9713702

N#Cc1cc(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)ccc1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 4/20 0.46
KMT2A Q03164 3/20 0.46
GAA P10253 2/20 0.46
HTT P42858 1/20 0.46
LMNA P02545 3/20 0.44
ALDH1A1 P00352 2/20 0.44
POLB P06746 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA3 P07451 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
CA5A P35218 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA13 Q8N1Q1 1/20 0.42
CA14 Q9ULX7 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL590624 0.88 KMT2A (0.51) VCAM1KMT2AGAAHTTLMNA
SCHEMBL590951 0.82 VCAM1 (0.50) VCAM1KMT2AGAAHTTLMNA
SCHEMBL698847 0.82 VCAM1 (0.66) VCAM1KMT2AGAALMNAALDH1A1
SCHEMBL589476 0.80 VCAM1 (0.48) VCAM1KMT2AGAAHTTLMNA
SCHEMBL20380311 0.77 KCNJ1 (0.51) VCAM1KMT2AGAAHTTPOLB
SCHEMBL11855965 0.76 CA2 (0.67) KMT2AGAAHTTLMNAALDH1A1
SCHEMBL3158508 0.76 CA2 (0.67) KMT2AGAAHTTLMNAALDH1A1
SCHEMBL11419996 0.76 CA2 (0.67) KMT2AGAAHTTLMNAALDH1A1
SCHEMBL9713754 0.76 MAPT (0.50) VCAM1KMT2AGAAHTTLMNA
Formic Acid SCHEMBL27641278 0.75 HPGD (0.44) VCAM1GAAHTTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084449-A Bactericides and antiprotozoa agents DR. KARL THOMAE GMBH (DE) 1992-01-28 US disclosed
US-4992430-A Anti-bacterial compositions comprising a substituted bis-(4-aminophenyl)-sulfone and a dihydro-folic acid reductase DR. KARL THOMAE GMBH (DE) 1991-02-12 US disclosed
US-4829058-A INHIBITORS OF BACTERIA, MYCOBACTERIA AND PLASMODIA DR. KARL THOMAE GMBH (DE) 1989-05-09 US disclosed
EP-0165422-B1 SUBSTITUTED BIS-(4-AMINOPHENYL)-SULPHONES, THEIR PREPARATION AND THEIR USE AS MEDICINES Dr. Karl Thomae GmbH (DE) 1988-03-09 EP disclosed
EP-0165422-A1 Substituted bis-(4-aminophenyl)-sulphones, their preparation and their use as medicines Dr. Karl Thomae GmbH (DE) 1985-12-27 EP disclosed