SCHEMBL9713827

SCHEMBL9713827

CC(C)C[C@@H](C(=O)N(C)C(=O)[C@@H](N)C(C)(C)C)C(CCCc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.39
MMP1 P03956 2/20 0.38
MMP3 P08254 2/20 0.38
MMP9 P14780 1/20 0.38
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MMP13 P45452 1/20 0.35
REN P00797 2/20 0.34
LTA4H P09960 1/20 0.34
ALOX5 P09917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714207 0.85 MMP1 (0.48) MMP1MMP3MMP9MMP13
SCHEMBL7837093 0.82 MMP1 (0.44) GRIK1MMP1MMP3MMP9MMP13
SCHEMBL7837095 0.82 MMP1 (0.44) GRIK1MMP1MMP3MMP9MMP13
SCHEMBL6987281 0.82 MMP3 (0.45) GRIK1MMP1MMP3MMP9REN
SCHEMBL6659520 0.82 MMP3 (0.45) GRIK1MMP1MMP3MMP9REN
SCHEMBL6943292 0.82 MMP3 (0.45) GRIK1MMP1MMP3MMP9REN
SCHEMBL6659518 0.82 MMP3 (0.45) GRIK1MMP1MMP3MMP9REN
SCHEMBL6943287 0.82 MMP3 (0.45) GRIK1MMP1MMP3MMP9REN
SCHEMBL7827850 0.79 MMP1 (0.46) GRIK1MMP1MMP3MMP9MMP13
SCHEMBL7853162 0.79 MMP1 (0.46) GRIK1MMP1MMP3MMP9MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497192-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-08-05 EP disclosed