SCHEMBL9715146

SCHEMBL9715146

C=CCC(C(=O)OCC)C(=O)c1cccc(F)c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.37
TSHR P16473 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
LMNA P02545 2/20 0.34
NLRP3 Q96P20 1/20 0.34
HCRTR2 O43614 2/20 0.33
CTSS P25774 1/20 0.33
HCRTR1 O43613 1/20 0.33
OPRK1 P41145 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KRAS P01116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9649781 0.86 KDM4E (0.44) TSHRALDH1A1TDP1SMN1; SMN2KDM4E
SCHEMBL9650664 0.82 SMN1; SMN2 (0.40) L3MBTL1TSHRALDH1A1MAPK1TDP1
SCHEMBL9650914 0.80 KMT2A (0.46) L3MBTL1TSHRALDH1A1MAPK1TDP1
SCHEMBL9647401 0.78 TDP1 (0.45) L3MBTL1TSHRALDH1A1TDP1SMN1; SMN2
SCHEMBL9649751 0.77 TSHR (0.42) L3MBTL1TSHRALDH1A1MAPK1TDP1
SCHEMBL9650272 0.76 LMNA (0.44) TSHRALDH1A1TDP1SMN1; SMN2NPC1
SCHEMBL9647521 0.76 KCNK3 (0.39) TSHRALDH1A1MAPK1TDP1KDM4E
SCHEMBL9647321 0.72 MEN1 (0.49) ALDH1A1MAPK1TDP1SMN1; SMN2NPC1
SCHEMBL27504359 0.71 NLRP3 (0.41) L3MBTL1TSHRALDH1A1MAPK1TDP1
SCHEMBL1825614 0.70 LMNA (0.43) L3MBTL1ALDH1A1MAPK1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266980-B1 PHARMACEUTICAL COMPOSITIONS, COMPRISING A 2,4-DIPHENYL-1,3-DIOXANE DERIVATIVE AND AN INHIBITOR OF THROMBOXANE A2 SYNTHESIS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-10-28 EP disclosed
EP-0201354-B1 2,4-DIPHENYL-1,3-DIOXANES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-09-19 EP disclosed
US-4908380-A Substituted 1,3-dioxane ether derivative; thromboxane A2 inhibitor IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-03-13 US disclosed
US-4895962-A THROMBOXANE A2 ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-01-23 US disclosed
US-4775685-A THROMBOXANE A-2 ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-10-04 US disclosed
EP-0201354-A2 2,4-Diphenyl-1,3-Dioxanes IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-11-12 EP disclosed