SCHEMBL9649751

SCHEMBL9649751

C=CCC(C(=O)OCC)C(=O)c1ccccc1CC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
TDP1 Q9NUW8 3/20 0.40
CYP3A4 P08684 1/20 0.40
L3MBTL1 Q9Y468 4/20 0.39
MAPK1 P28482 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
MMP8 P22894 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
RECQL P46063 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 2/20 0.38
LMNA P02545 2/20 0.37
PIN1 Q13526 1/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9647401 0.87 TDP1 (0.45) TSHRTDP1CYP3A4L3MBTL1MEN1
SCHEMBL9650318 0.85 CYP2C19 (0.46) CYP3A4MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL9650272 0.85 LMNA (0.44) TSHRTDP1CYP3A4MEN1KMT2A
SCHEMBL9649781 0.85 KDM4E (0.44) TSHRTDP1CYP3A4MEN1KMT2A
SCHEMBL9650914 0.84 KMT2A (0.46) TSHRTDP1L3MBTL1MAPK1MEN1
SCHEMBL9647521 0.82 KCNK3 (0.39) TSHRTDP1CYP3A4MAPK1MEN1
SCHEMBL9647321 0.81 MEN1 (0.49) TDP1MAPK1MEN1KMT2ANPC1
SCHEMBL9715146 0.77 L3MBTL1 (0.37) TSHRTDP1L3MBTL1MAPK1KMT2A
SCHEMBL1825614 0.76 LMNA (0.43) L3MBTL1MAPK1MEN1KMT2AMMP8
SCHEMBL286 0.75 SLC6A3 (0.51) TSHRTDP1L3MBTL1MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5166377-A Thromboxane A2 antagonist as coagulants or vasoconstrictors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-11-24 US disclosed
US-4745198-A CARDIOVASCULAR DISORDERS, BRONCHODILATOR AGENTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-05-17 US disclosed
EP-0094239-B1 1,3-DIOXAN-5-YLALKENOIC ACIDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-07-15 EP disclosed
US-4567197-A THORMBOXANE A2 ANTAGONISTS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-01-28 US disclosed
EP-0094239-A2 1,3-Dioxan-5-ylalkenoic acids IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-16 EP disclosed