SCHEMBL971766

SCHEMBL971766

CCOC(=O)c1cs[c]n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.50
RAB9A P51151 6/20 0.50
NPC1 O15118 5/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 2/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.43
GAA P10253 3/20 0.43
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
GABRA2 P47869 2/20 0.41
GABRB2 P47870 2/20 0.41
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743243 0.81
SCHEMBL4474111 0.72 CNR1 (0.39) RAB9ANPC1ALDH1A1KMT2ACYP2C19
SCHEMBL969213 0.71 MEN1 (0.51) MAPTALDH1A1CYP1A2MEN1KMT2A
SCHEMBL1444391 0.71
SCHEMBL17028993 0.70 ALDH1A1 (0.46) MAPTRAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL971952 0.70 ALDH1A1 (0.44) MAPTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL243257 0.70 MAPT (0.50) MAPTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL13144514 0.70 MAPT (0.70) MAPTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL3702158 0.70 MAPT (0.61) MAPTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL914552 0.70 RAB9A (0.68) MAPTRAB9ANPC1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 221 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118344265-A Amide compound and preparation method and application thereof 河北大学 2024-07-16 CN claimed
EP-2668183-B1 IL17 AND IFN-GAMMA INHIBITION FOR THE TREATMENT OF AUTOIMMUNE INFLAMMATION 4SC DISCOVERY GMBH (DE) 2017-11-01 EP claimed
US-9238658-B2 Substituted piperidinyl-carboxamide derivatives useful as SCD 1 inhibitors JANSSEN PHARMACEUTICA NV (BE) 2016-01-19 US claimed
CN-103459385-B IL17 and the IFN-γ being used for the treatment of autoimmune inflammation suppresses 4SC DISCOVERY GMBH (DE) 2015-08-05 CN claimed
CN-104206385-A Use of amine compound as bactericide SINOCHEM CORP 2014-12-17 CN claimed
US-20140364393-A1 SUBSTITUTED PIPERIDINYL-CARBOXAMIDE DERIVATIVES USEFUL AS SCD 1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2014-12-11 US claimed
CN-103459385-A IL17 and IFN-[gamma] inhibition for the treatment of autoimmune inflammation 4SC DISCOVERY GMBH 2013-12-18 CN claimed
WO-2013085954-A1 SUBSTITUTED PIPERIDINYL-CARBOXAMIDE DERIVATIVES USEFUL AS SCD 1 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2013-06-13 WO claimed
CN-102942565-A 3,4-dichloro isothiazole derivatives, their preparation method and application JIANGXI TIANREN ECOLOGY CO LTD 2013-02-27 CN claimed
US-8354436-B2 IL17 and IFN-gamma inhibition for the treatment of autoimmune inflammation 4SC DISCOVERY GMBH (DE) 2013-01-15 US claimed
US-6262103-B1 ALZHEIMER'S DISEASE. MERCK SHARP & DOHME LIMITED (GB) 2001-07-17 US claimed
JP-2001503408-A 2001-03-13 JP claimed
EP-0937072-A1 THIENYLCYCLOHEXANONE DERIVATIVES AS LIGANDS OF THE GABA A? $g(a)5 RECEPTOR SUBTYPE MERCK SHARP & DOHME LTD. (GB) 1999-08-25 EP claimed
WO-1998018792-A1 THIENYLCYCLOHEXANONE DERIVATIVES AS LIGANDS OF THE GABAA α5 RECEPTOR SUBTYPE MERCK SHARP & DOHME LIMITED (GB) 1998-05-07 WO claimed
US-5158598-A Insecticides, miticides, and nematocides; nonphytotoxic BASF AKTIENGESELLSCHAFT (DE) 1992-10-27 US claimed
EP-0248735-B1 2-Thiazolyl imidazo [1,2-a] pyrimidines and their salts, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1990-05-23 EP claimed
US-4925846-A COGNITION ACTIVATORS, TRANQUILIZERS, DIETETICS ROUSSEL UCLAF (FR) 1990-05-15 US claimed
US-4829053-A Amino acid derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-05-09 US claimed
EP-0248735-A1 2-Thiazolyl imidazo [1,2-a] pyrimidines and their salts, process for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1987-12-09 EP claimed
US-4243669-A ANTICOAGULANTS BEECHAM GROUP LIMITED (GB) 1981-01-06 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140364393-A1 SUBSTITUTED PIPERIDINYL-CARBOXAMIDE DERIVATIVES USEFUL AS SCD 1 INHIBITORS SCD, SCD5, FASN MAPT 4508/4885RAB9A 2991/4885NPC1 120/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.