SCHEMBL972258

SCHEMBL972258

CC1CN(S(=O)(=O)c2ccc(NC(=O)c3c(Cl)cccc3NS(=O)(=O)c3ccc(Cl)cc3)cc2)CC(C)O1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.55
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
ALDH1A1 P00352 3/20 0.53
RXFP1 Q9HBX9 1/20 0.51
DDIT3 P35638 1/20 0.49
LMNA P02545 3/20 0.48
NPSR1 Q6W5P4 2/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
USP2 O75604 2/20 0.48
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
GPR27 Q9NS67 2/20 0.47
CXCR2 P25025 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL491583 0.86 ALDH1A1 (0.55) MEN1KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL491976 0.83 THRB (0.59) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491991 0.83 THRB (0.59) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491990 0.83 THRB (0.59) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491977 0.83 THRB (0.59) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL971693 0.83 LMNA (0.52) MEN1KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL491687 0.80 THRB (0.55) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491688 0.80 THRB (0.55) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491849 0.79 THRB (0.54) THRBMEN1KMT2AALDH1A1RXFP1
SCHEMBL491847 0.79 THRB (0.54) THRBMEN1KMT2AALDH1A1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207541-B1 USE OF SULFONYL-SUBSTITUTED 2-SULFONYLAMINOBENZOIC ACID N-PHENYLAMIDES IN THE TREATMENT OF PAIN SANOFI AVENTIS DEUTSCHLAND (DE) 2014-10-29 EP disclosed
US-8518998-B2 Use of sulfonyl-substituted 2-sulfonylaminobenzoic acid N-phenylamides in the treatment of pain SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2013-08-27 US disclosed
CN-101815514-B Use of sulfonyl-substituted 2-sulfonylaminobenzoic acid N-phenylamides in the treatment of pain SANOFI AVENTIS DEUTSCHLAND 2012-05-09 CN disclosed
US-20110021505-A1 Use of sulfonyl-substituted 2-sulfonylaminobenzoic acid N-phenylamides in the treatment of pain SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2011-01-27 US disclosed
CN-101815514-A Use of sulfonyl-substituted 2-sulfonylaminobenzoic acid N-phenylamides in the treatment of pain SANOFI AVENTIS DEUTSCHLAND 2010-08-25 CN disclosed
EP-2207541-A1 USE OF SULFONYL-SUBSTITUTED 2-SULFONYLAMINOBENZOIC ACID N-PHENYLAMIDES IN THE TREATMENT OF PAIN Sanofi-Aventis Deutschland GmbH (DE) 2010-07-21 EP disclosed
WO-2009043495-A1 USE OF SULFONYL-SUBSTITUTED 2-SULFONYLAMINOBENZOIC ACID N-PHENYLAMIDES IN THE TREATMENT OF PAIN SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2009-04-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021505-A1 Use of sulfonyl-substituted 2-sulfonylaminobenzoic acid N-phenylamides in the treatment of pain SCN1A, SCN2A, CACNA1A THRB 1294/4885MEN1 3830/4885KMT2A 568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.