SCHEMBL9722607

SCHEMBL9722607

[O-][S+](CCCCCl)Cc1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CHRNA7 P36544 2/20 0.39
HRH1 P35367 2/20 0.38
CHRNB2 P17787 3/20 0.38
CHRNA4 P43681 3/20 0.38
CHRM2 P08172 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
CYP2C19 P33261 1/20 0.36
TBXAS1 P24557 1/20 0.36
BTN3A1 O00481 1/20 0.36
FDPS P14324 1/20 0.36
PDE3A Q14432 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9626044 0.80 CALM1 (0.31) TDP1
SCHEMBL9270295 0.79 NAPRT (0.43) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL27287431 0.77 CYP2C9 (0.38) CYP1A2CYP2D6TDP1HRH1CHRNB2
SCHEMBL12854098 0.75 CHRNB2 (0.49) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL10333077 0.74 CALM1 (0.32) CYP1A2CYP2D6TDP1HRH1CHRM2
SCHEMBL826569 0.74 TDP1 (0.67) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL742233 0.73 HRH1 (0.68) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL740922 0.73 HRH1 (0.68) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL10350863 0.73 HRH1 (0.68) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1
SCHEMBL10349750 0.73 HRH1 (0.68) CYP2A6CYP1A2CYP2D6TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120852-A Contacting an alkyl isothiocyanate with an anionized sulfoxide RHONE-POULENC SANTE (FR) 1992-06-09 US disclosed
US-4751234-A Certain N-alkyl-2-[(quinolin-3-yl)-tetrahydro-pyran or furan]-2-carbothiamide 1-oxide derivatives useful for treating hypertension RHONE-POULENC SANTE (FR) 1988-06-14 US disclosed
US-4568682-A Certain N-lower-alkyl-2-(pyridin-3yl)-tetrahydrothiophene or tetrahydrothiopyran-2-carbothioamide-1-oxides having anti-hypertensive activity RHONE-POULENC SANTE (FR) 1986-02-04 US disclosed