SCHEMBL9724160

SCHEMBL9724160

O=c1cc(O)c2cc(-c3ccccc3)ccc2[nH]1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.64
ALDH1A1 P00352 1/20 0.64
TNKS2 Q9H2K2 2/20 0.55
BRD4 O60885 2/20 0.53
HTT P42858 2/20 0.53
HPGD P15428 1/20 0.53
MAPK1 P28482 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
CDK4 P11802 1/20 0.49
CCND1 P24385 1/20 0.49
AR P10275 1/20 0.48
KDM5A P29375 1/20 0.45
HDAC4 P56524 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
MPL P40238 1/20 0.44
FEN1 P39748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11705503 0.81 TNKS2 (0.76) KDM4EALDH1A1TNKS2BRD4HTT
SCHEMBL1193735 0.78 KDM4E (1.00) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL29624606 0.78 KDM4E (1.00) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL1771872 0.76 AR (0.61) TNKS2AR
SCHEMBL19041639 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL149685 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL29386403 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL3365890 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL30300831 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD
SCHEMBL17154708 0.76 CDK4 (0.57) KDM4EALDH1A1TNKS2HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed