SCHEMBL9724254

SCHEMBL9724254

Cc1cc(C#N)c2cc(CBr)ccc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRB O95718 1/20 0.38
ESR1 P03372 1/20 0.38
ESRRA P11474 1/20 0.38
ESR2 Q92731 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
TSHR P16473 2/20 0.38
MAPK1 P28482 1/20 0.38
PKM P14618 1/20 0.37
KDM4E B2RXH2 4/20 0.36
GAA P10253 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 4/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
LMNA P02545 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6765981 0.83 ESR1 (0.39) ESRRBESR1ESRRAESR2L3MBTL1
SCHEMBL25174784 0.80 ALDH1A1 (0.48) ESRRBESR1ESRRAESR2KDM4E
SCHEMBL30368885 0.80 ALDH1A1 (0.48) ESRRBESR1ESRRAESR2KDM4E
SCHEMBL6766208 0.79 LMNA (0.56) ESRRBESR1ESRRAESR2L3MBTL1
SCHEMBL12638631 0.79 CYP1A2 (0.52) MAPK1KDM4EGAAALDH1A1CYP3A4
SCHEMBL9724225 0.78 ALDH1A1 (0.39) ESRRBESR1ESRRAESR2L3MBTL1
SCHEMBL9380126 0.76 LMNA (0.62) L3MBTL1KDM4EGAARXFP1ALDH1A1
SCHEMBL9724145 0.76 KDM4E (0.38) L3MBTL1TSHRKDM4EGAAALDH1A1
SCHEMBL9724218 0.74 DOT1L (0.49) ESR1ESR2KDM4EALDH1A1KMT2A
SCHEMBL9724298 0.74 MAPT (0.40) L3MBTL1KDM4EGAANPSR1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed