SCHEMBL9724145

SCHEMBL9724145

Cc1cc(O)c2cc(CBr)ccc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.38
ALDH1A1 P00352 7/20 0.38
HPGD P15428 4/20 0.38
GAA P10253 2/20 0.38
GLA P06280 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
KMT2A Q03164 4/20 0.38
RAD52 P43351 3/20 0.38
POLB P06746 3/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
ALPL P05186 1/20 0.37
ALPG P10696 1/20 0.37
PLAA Q9Y263 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 2/20 0.37
MEN1 O00255 3/20 0.37
GNG2 P59768 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12638631 0.83 CYP1A2 (0.52) KDM4EALDH1A1HPGDGAACYP3A4
SCHEMBL9724225 0.81 ALDH1A1 (0.39) KDM4EALDH1A1HPGDGAACYP3A4
SCHEMBL9380126 0.80 LMNA (0.62) KDM4EALDH1A1HPGDGAACYP3A4
SCHEMBL9724298 0.78 MAPT (0.40) KDM4EALDH1A1HPGDGAACYP3A4
SCHEMBL9724218 0.78 DOT1L (0.49) KDM4EALDH1A1HPGDKMT2APOLB
SCHEMBL4966064 0.77 ALDH1A1 (0.55) KDM4EALDH1A1GAACYP2C19KMT2A
SCHEMBL29923741 0.77 ALDH1A1 (0.55) KDM4EALDH1A1GAACYP2C19KMT2A
SCHEMBL3760247 0.77 LMNA (0.61) KDM4EALDH1A1GAACYP3A4CYP2C19
SCHEMBL9724254 0.76 ESRRB (0.38) KDM4EALDH1A1HPGDGAACYP3A4
SCHEMBL4748554 0.74 POLB (0.53) KDM4EALDH1A1KMT2APOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed