SCHEMBL9724306

SCHEMBL9724306

COc1cc(C)nc2ccc(C)cc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.59
LMNA P02545 1/20 0.58
DOT1L Q8TEK3 1/20 0.55
TERT O14746 2/20 0.52
GAA P10253 1/20 0.52
KCNH2 Q12809 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
PKM P14618 1/20 0.46
CYP1A2 P05177 1/20 0.46
ACHE P22303 1/20 0.45
MITF O75030 1/20 0.45
MAPT P10636 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PTPN11 Q06124 1/20 0.44
ALDH1A1 P00352 2/20 0.44
RAD52 P43351 1/20 0.44
NQO2 P16083 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699246 0.84 KDM4E (0.49) KDM4ELMNADOT1LTERTGAA
SCHEMBL4219099 0.84 LMNA (0.61) KDM4ELMNADOT1LGAAKCNH2
SCHEMBL11039427 0.82 CRHR1 (0.52) LMNADOT1LTERTKCNH2MAPT
SCHEMBL9381975 0.82 BACE1 (0.49) KDM4ELMNAGAAKMT2AMEN1
SCHEMBL5848248 0.82 DOT1L (0.52) KDM4ELMNADOT1LTERTGAA
SCHEMBL2534913 0.82 LMNA (0.50) KDM4ELMNADOT1LGAAKMT2A
SCHEMBL19689623 0.82 ESR1 (0.49) KDM4ELMNADOT1LGAAKCNH2
SCHEMBL24003870 0.80 DOT1L (0.50) KDM4EDOT1LTERTGAAL3MBTL1
SCHEMBL29324282 0.80 DOT1L (0.53) KDM4ELMNADOT1LTERTGAA
SCHEMBL266444 0.79 LMNA (0.64) KDM4ELMNADOT1LGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed