SCHEMBL9724927

SCHEMBL9724927

O=C(NCCCCN1CCN(c2cccc(C(F)(F)F)n2)CC1)c1ccc(F)cc1

nearest known ligand 0.87

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.87
DRD3 P35462 8/20 0.62
HTR2A P28223 5/20 0.62
DRD2 P14416 6/20 0.60
DRD4 P21917 4/20 0.60
ADRA1A P35348 3/20 0.60
ADRA1D P25100 2/20 0.60
ADRA1B P35368 2/20 0.60
CCR3 P51677 1/20 0.52
HTR2C P28335 2/20 0.51
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9725005 0.93 HTR1A (1.00) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL9725016 0.92 HTR1A (0.73) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL9725045 0.85 HTR1A (0.84) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL14761668 0.82 HTR1A (0.70) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL14761321 0.81 DRD3 (0.77) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL9725055 0.80 HTR1A (0.64) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL27726458 0.78 HTR1A (0.73) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL9725026 0.78 HTR1A (0.70) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL14761844 0.77 DRD3 (0.72) HTR1ADRD3HTR2ADRD2DRD4
SCHEMBL9725141 0.77 HTR1A (0.66) HTR1ADRD3HTR2ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135931-A Antidepressants, psychological disorders, nervous system disorders AKZO N.V. (NL) 1992-08-04 US disclosed
EP-0462638-A1 Pyridinylpiperazine derivatives Akzo Nobel N.V. (NL) 1991-12-27 EP disclosed