SCHEMBL9725005

SCHEMBL9725005

O=C(NCCN1CCN(c2cccc(C(F)(F)F)n2)CC1)c1ccc(F)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 1.00
DRD2 P14416 1/20 0.55
DRD4 P21917 1/20 0.54
HTR1D P28221 1/20 0.54
ADRA1A P35348 1/20 0.54
HTR2B P41595 1/20 0.54
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HTR2A P28223 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9724927 0.93 HTR1A (0.87) HTR1ADRD2DRD4ADRA1AHTR2B
SCHEMBL9725045 0.92 HTR1A (0.84) HTR1ADRD2DRD4HTR2BMAPT
SCHEMBL9725016 0.84 HTR1A (0.73) HTR1ADRD2DRD4ADRA1AHTR2A
SCHEMBL27726458 0.84 HTR1A (0.73) HTR1ADRD2DRD4HTR2BHTR2A
SCHEMBL9725026 0.82 HTR1A (0.70) HTR1ADRD2DRD4HTR2BHTR2A
SCHEMBL14761329 0.81 HTR1A (0.67) HTR1ADRD2DRD4CYP1A2CYP3A4
SCHEMBL9725141 0.80 HTR1A (0.66) HTR1ADRD2DRD4ADRA1AHTR2B
SCHEMBL14761918 0.79 HTR1A (0.66) HTR1ADRD4MAPTHSD17B10HTR2A
SCHEMBL9724944 0.78 HTR1A (0.64) HTR1ADRD2DRD4
SCHEMBL9725055 0.78 HTR1A (0.64) HTR1ADRD2DRD4HTR2BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135931-A Antidepressants, psychological disorders, nervous system disorders AKZO N.V. (NL) 1992-08-04 US claimed
EP-0462638-A1 Pyridinylpiperazine derivatives Akzo Nobel N.V. (NL) 1991-12-27 EP claimed
US-5135931-A Antidepressants, psychological disorders, nervous system disorders AKZO N.V. (NL) 1992-08-04 US disclosed
EP-0462638-A1 Pyridinylpiperazine derivatives Akzo Nobel N.V. (NL) 1991-12-27 EP disclosed