SCHEMBL9726216

SCHEMBL9726216

O=C(c1ccc(F)cc1)C1CCN(CCCN2c3ccccc3-c3ccccc3S2(=O)=O)CC1

nearest known ligand 0.75

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.56
KDM4E B2RXH2 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
HTR2C P28335 5/20 0.54
HTR7 P34969 2/20 0.54
HTR6 P50406 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9667623 0.87 HTR2A (0.60) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9757250 0.85 HTR7 (0.66) HTR2AHTR2CHTR7HTR6
SCHEMBL6995331 0.82 HTR2A (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6991299 0.80 HTR2A (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6991294 0.80 HTR2A (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9726227 0.79 DRD2 (0.72) HTR2AHTR2CHTR7HTR6
SCHEMBL9757356 0.79 HTR2A (0.57) HTR2AHTR2CHTR7HTR6
SCHEMBL6995673 0.76 HTR2A (0.58) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL11799453 0.75 HTR2A (0.62) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL7816022 0.75 HTR2C (0.56) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130313-A Central nervous system disorders, cardiovascular disorders or gastrointestinal disorders RHONE-POULENC SANTE (FR) 1992-07-14 US disclosed