SCHEMBL9726400

SCHEMBL9726400

COc1ccc(CNc2cnn(C(C)C)c(=O)c2C)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 8/20 0.62
KDM4C Q9H3R0 1/20 0.51
NPC1 O15118 1/20 0.45
PKM P14618 1/20 0.45
RAB9A P51151 1/20 0.45
APLNR P35414 1/20 0.45
TSHR P16473 6/20 0.44
LMNA P02545 2/20 0.44
HPGD P15428 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ERBB2 P04626 1/20 0.44
PRKACA P17612 1/20 0.44
RPS6KB1 P23443 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
IRAK1 P51617 1/20 0.44
RPS6KA3 P51812 1/20 0.44
ROCK1 Q13464 1/20 0.44
CDC42BPA Q5VT25 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726419 0.88 PDE9A (0.61) PDE9AKDM4CNPC1PKMRAB9A
SCHEMBL10601720 0.88 PDE9A (0.61) PDE9AKDM4CNPC1PKMRAB9A
SCHEMBL9726712 0.87 PDE9A (0.60) PDE9AKDM4CNPC1PKMRAB9A
SCHEMBL9726658 0.85 PDE9A (0.58) PDE9AKDM4CNPC1PKMRAB9A
SCHEMBL9726564 0.83 PDE9A (0.58) PDE9AMEN1KMT2AGAAMAPT
SCHEMBL9726447 0.80 PDE9A (0.61) PDE9AKDM4CNPC1PKMRAB9A
SCHEMBL9726518 0.78 BRD4 (0.51) PDE9AKDM4CNPC1RAB9ASMN1; SMN2
SCHEMBL16981660 0.76 PDE9A (1.00) PDE9A
SCHEMBL9726397 0.76 KDM4E (0.45) PDE9ATSHRLMNAHPGDSMN1; SMN2
SCHEMBL9726861 0.74 POLB (0.41) PDE9ATSHRLMNAHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed