SCHEMBL9726447

SCHEMBL9726447

COc1ccc(CNc2cnn(C(C)C)c(=O)c2)c(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 5/20 0.61
ERBB2 P04626 1/20 0.48
PRKACA P17612 1/20 0.48
RPS6KB1 P23443 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
IRAK1 P51617 1/20 0.48
RPS6KA3 P51812 1/20 0.48
ROCK1 Q13464 1/20 0.48
CDC42BPA Q5VT25 1/20 0.48
AURKB Q96GD4 1/20 0.48
CSNK1G3 Q9Y6M4 1/20 0.48
KDM4C Q9H3R0 1/20 0.47
APLNR P35414 1/20 0.47
NPC1 O15118 1/20 0.47
PKM P14618 1/20 0.47
RAB9A P51151 1/20 0.47
GAA P10253 2/20 0.45
TP53 P04637 1/20 0.45
FGFR3 P22607 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726400 0.80 PDE9A (0.62) PDE9AERBB2PRKACARPS6KB1GSK3A
SCHEMBL9726419 0.79 PDE9A (0.61) PDE9AERBB2PRKACARPS6KB1GSK3A
SCHEMBL10601720 0.79 PDE9A (0.61) PDE9AERBB2PRKACARPS6KB1GSK3A
SCHEMBL9726712 0.78 PDE9A (0.60) PDE9AERBB2PRKACARPS6KB1GSK3A
SCHEMBL9726658 0.77 PDE9A (0.58) PDE9AERBB2PRKACARPS6KB1GSK3A
SCHEMBL16981660 0.76 PDE9A (1.00) PDE9A
SCHEMBL24851746 0.75 PDE9A (0.56) PDE9ANPC1PKMRAB9AGAA
SCHEMBL30162264 0.75 PDE9A (0.56) PDE9ANPC1PKMRAB9AGAA
SCHEMBL27948920 0.73 APLNR (0.69) ERBB2PRKACARPS6KB1GSK3AGSK3B
SCHEMBL855657 0.71 APLNR (0.58) ERBB2PRKACARPS6KB1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed