SCHEMBL9726419

SCHEMBL9726419

COc1ccc(CNc2cnn(C(C)C)c(=O)c2Cl)c(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 6/20 0.61
KDM4C Q9H3R0 2/20 0.50
TSHR P16473 4/20 0.45
ALDH1A1 P00352 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
CYP2C9 P11712 3/20 0.45
CYP2C19 P33261 3/20 0.45
HIF1A Q16665 2/20 0.45
HSD17B10 Q99714 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
BPTF Q12830 1/20 0.45
P2RX3 P56373 1/20 0.45
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
APLNR P35414 1/20 0.44
ERBB2 P04626 1/20 0.43
PRKACA P17612 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726400 0.88 PDE9A (0.62) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL10601720 0.87 PDE9A (0.61) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL9726712 0.86 PDE9A (0.60) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL9726658 0.85 PDE9A (0.58) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL9726824 0.84 PDE9A (0.49) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL9726598 0.81 BPTF (0.52) PDE9ATSHRALDH1A1TDP1BPTF
SCHEMBL9726869 0.80 BPTF (0.49) PDE9ABPTFBRD4KAT2BLMNA
SCHEMBL10681057 0.80 BPTF (0.42) PDE9ABPTFRAB9AGAAKAT2B
SCHEMBL9726447 0.79 PDE9A (0.61) PDE9AKDM4CTSHRALDH1A1CYP1A2
SCHEMBL9726613 0.78 BPTF (0.49) PDE9ATSHRALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US claimed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP claimed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP claimed
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed