SCHEMBL9726458

SCHEMBL9726458

O=C(c1c(Cl)cccc1Cl)c1c(Cl)cccc1Cl

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.67
FEN1 P39748 1/20 0.50
HPGD P15428 2/20 0.48
NPC1 O15118 1/20 0.48
GLA P06280 1/20 0.48
DOT1L Q8TEK3 2/20 0.47
TSHR P16473 2/20 0.46
AKR1B1 P15121 1/20 0.46
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
JAK2 O60674 1/20 0.45
CYP3A4 P08684 1/20 0.45
JAK1 P23458 1/20 0.45
TYK2 P29597 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP2A6 P11509 1/20 0.43
RORC P51449 1/20 0.42
GAA P10253 1/20 0.42
PBRM1 Q86U86 1/20 0.42
DPP4 P27487 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1042856 0.85 ALDH1A1 (0.59) ALDH1A1FEN1DOT1LTSHRCES2
SCHEMBL11850279 0.83 SRD5A2 (0.56) ALDH1A1HPGDDOT1LTSHRCES2
SCHEMBL2876974 0.83 GAA (0.58) ALDH1A1HPGDCES2CES1JAK2
SCHEMBL611393 0.81 MAPK1 (0.59) ALDH1A1HPGDDOT1LCES2GAA
SCHEMBL80183 0.80 ALDH1A1 (0.64) ALDH1A1FEN1HPGDNPC1GLA
SCHEMBL19998299 0.80 ALDH1A1 (0.64) ALDH1A1FEN1HPGDNPC1GLA
SCHEMBL103586 0.80 ALDH1A1 (1.00) ALDH1A1FEN1HPGDNPC1GLA
SCHEMBL80182 0.80 ALDH1A1 (0.64) ALDH1A1FEN1HPGDNPC1GLA
SCHEMBL1594842 0.79 ALDH1A1 (0.45) ALDH1A1FEN1HPGDNPC1GLA
SCHEMBL9515912 0.79 ALDH1A1 (0.45) ALDH1A1FEN1HPGDNPC1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103748076-A ROR gamma T inhibitors MERCK SHARP & DOHME 2014-04-23 CN claimed
CN-104940202-B Inhibitors of influenza viruses replication 沃泰克斯药物股份有限公司 2018-10-16 CN disclosed
CN-107771178-A Synthesis of heterocyclic compounds 普莱希科公司 2018-03-06 CN disclosed
CN-105531274-A Keto-imidazopyridine derivatives as rorc modulators HOFFMANN LA ROCHE 2016-04-27 CN disclosed
CN-103748076-A ROR gamma T inhibitors MERCK SHARP & DOHME 2014-04-23 CN disclosed
CN-1743355-A Sulfonic group-containing polyarylene block copolymer, process for production thereof, solid polymer electrolyte and proton conductive membrane JSR CORP (JP) 2006-03-08 CN disclosed
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed