SCHEMBL9726477

SCHEMBL9726477

CCOc1cccc(CNc2cnn(C(C)C)c(=O)c2CC)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 5/20 0.48
PDE1A P54750 5/20 0.43
PDE1B Q01064 5/20 0.43
PDE1C Q14123 5/20 0.43
APAF1 O14727 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
BRD4 O60885 1/20 0.40
BRD9 Q9H8M2 1/20 0.40
BPTF Q12830 1/20 0.39
GRM2 Q14416 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
ROCK2 O75116 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ROCK1 Q13464 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726499 0.92 PDE9A (0.47) PDE9APDE1APDE1BPDE1CAPAF1
SCHEMBL9726558 0.88 PDE9A (0.49) PDE9APDE1APDE1BPDE1CAPAF1
SCHEMBL9726528 0.88 BRD4 (0.52) PDE9APDE1APDE1BPDE1CAPAF1
SCHEMBL9726483 0.85 BRD4 (0.41) PDE9ABRD4BRD9BPTFGRM2
SCHEMBL9726486 0.82 PDE9A (0.57) PDE9AGRM2GAAMAPT
SCHEMBL9726540 0.82 KDM4E (0.44) PDE9AAPAF1L3MBTL1SMN1; SMN2GAA
SCHEMBL9726516 0.79 PDE9A (0.56) PDE9APDE1APDE1BPDE1CBPTF
SCHEMBL9726508 0.78 BRD4 (0.52) PDE9AL3MBTL1BRD4BRD9BPTF
SCHEMBL9726443 0.77 BACE1 (0.43) PDE9AAPAF1L3MBTL1BRD4BRD9
SCHEMBL9726399 0.75 BRD4 (0.49) PDE9ABRD4BRD9BPTFGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed