SCHEMBL9726486

SCHEMBL9726486

CCCc1c(NCc2cccc(OC)c2)cnn(C(C)C)c1=O

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 6/20 0.57
GRM2 Q14416 2/20 0.49
ABCB1 P08183 3/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
ALDH1A1 P00352 3/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 1/20 0.43
GAA P10253 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
EGFR P00533 1/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
CRHBP P24387 1/20 0.41
KMT2A Q03164 1/20 0.41
CRHR2 Q13324 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726499 0.91 PDE9A (0.47) PDE9AGRM2
SCHEMBL9726473 0.87 PDE9A (0.54) PDE9AGRM2
SCHEMBL9726658 0.83 PDE9A (0.58) PDE9AALDH1A1TSHRRAB9AGAA
SCHEMBL9726477 0.82 PDE9A (0.48) PDE9AGRM2GAAMAPT
SCHEMBL9726516 0.78 PDE9A (0.56) PDE9AGRM2
SCHEMBL9726558 0.77 PDE9A (0.49) PDE9AGRM2
SCHEMBL9726528 0.76 BRD4 (0.52) PDE9AGRM2ALDH1A1GAAMAPT
SCHEMBL9726712 0.74 PDE9A (0.60) PDE9AALDH1A1TSHRRAB9AGAA
SCHEMBL16981661 0.73 PDE9A (1.00) PDE9A
SCHEMBL9726540 0.73 KDM4E (0.44) PDE9AALDH1A1TSHRGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098900-A Reducing contractions in smooth muscles NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1992-03-24 US disclosed
EP-0186817-B1 3(2H)PYRIDAZINONE, PROCESS FOR ITS PREPARATION AND ANTI-ALLERGIC AGENT CONTAINING IT NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1989-08-02 EP disclosed
EP-0186817-A1 3(2H)pyridazinone, process for its preparation and anti-allergic agent containing it NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1986-07-09 EP disclosed